Phase 2: active escalation (weeks 8 to 24) As doses increase toward the therapeutic range of 8 to 12 mg, heart rate effects become more apparent
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This includes people with kidney and liver disease, those with diseases related to the blood, and women who are pregnant
Since HRAS mutations are found in Spitz nevus, but not in Spitzoid melanoma, HRAS may be used as a diagnostic test to help differentiate between these two lesions [114, 115]